Synthesis of 5-(2-Allylamino-1-hydroxyalkyl)-8-hydroxycarbostyrils, New β-Adrenoceptor Stimulants

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概要

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• A series of 5-(2-allylamino-1-hydroxyalkyl)-8-hydroxycarbostyrils (4) was synthesized. The β-adrenoceptor stimulant activities of erythro-5-(2-allylamino-1-hydroxypropyl)-8-hydroxycarbostyril (4b) in anesthetized dogs were determined.

• 社団法人日本薬学会の論文
• 1980-12-25

著者

• 田村 恭光

  Faculty Of Pharmaceutical Sciences Osaka University

• 楊 永雄

  Tokushima Research Institute, Otsuka Pharmaceutical Co., Ltd.,

• 中川 量之

  Laboratories of Medicinal Chemistry

• 吉崎 司郎

  (present Address)bio-center Nkk Corporation

• 楊 永雄

  Tokushima Research Institute Otsuka Pharmaceutical Co. Ltd.

• 中川 量之

  Laboratories Of Medicinal Chemistry Tokushima Research Institute Otsuka Pharmaceutical Co. Ltd.

• 田村 恭光

  Faculty of Pharmaceutical Sciences, Osaka University

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