Reaction of Benzo [b] furan and 1-Acylindoles with Iodine Azide
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概要
- 論文の詳細を見る
Reaction of benzo [b] furan with iodine azide gives in high yield a mixture of cis-and trans-2,3-diazido-2,3-dihydrobenzo [b] furans, both of which, upon treatment with alkali, are converted to 3-azidobenzo [b] furan. Similar reaction of 1-benzoyl-and 1-tosyl-indoles with iodine azide affords high yields of cis-and trans-1-benzoyl-and 1-tosyl-2,3-diazidoindolines. Stereochemical assignment of the adducts is made on the basis of nuclear magnetic resonance spectroscopy.
- 社団法人日本薬学会の論文
- 1978-11-25
著者
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田村 恭光
Faculty Of Pharmaceutical Sciences Osaka University
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千 文宇
Faculty of Pharmaceutical Sciences, Osaka University
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権 順度
Faculty of Pharmaceutical Sciences, Osaka University
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池田 正澄
Faculty of Pharmaceutical Sciences, Osaka University
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権 順度
Faculty Of Pharmaceutical Sciences Osaka University
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池田 正澄
Kyoto Pharmaceutical University
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千 文宇
Faculty Of Pharmaceutical Sciences Osaka University
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サイド モハメド
Faculty of Pharmaceutical Sciences, Osaka University
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岡田 智子
Faculty of Pharmaceutical Sciences, Osaka University
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サイド モハメド
Faculty Of Pharmaceutical Sciences Osaka University
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岡田 智子
Faculty Of Pharmaceutical Sciences Osaka University
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