Potential Anti-cancer Agents. II. 4-Azidoquinoline and 4-Azidopyridine Derivatives.
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概要
- 論文の詳細を見る
4-Azidoquinoline (VII) and its N-oxide (IV) were prepared from the corresponding hydrazino compounds (VI and III) with sodium nitrite and also from chloro compounds (II) with sodium azide. Similarly, 4-azidopyridine 1-oxide and 4-azido-2-picoline were obtained. The addition reaction of their azido group to propargyl alcohol, photolysis, and thermal decomposition were examined.
- 公益社団法人日本薬学会の論文
- 1961-02-25
著者
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板井 孝信
Showa College of Pharmaceutical Sciences
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板井 孝信
National Institute of Hygienic Sciences
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神谷 庄造
National Institute Of Hygienic Sciences
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- Synthesis, Chemical Properties and Mutagenicity of 1,6- and 3,6-Dinitrobenzo[a]pyrenes
- Synthesis of Antitumor Pyridine and Pyridazine N-Oxides having (2-Chloroethyl) nitrosoureidomethyl and Bis (2-chloroethyl)-aminomethyl Groups
- Antitumor Activity of 4-Nitropyridazine 1-Oxides and Related Compounds for AH-13
- Mutagenic and Prophage-inducing Activities of 1-Alkyl-3-nitrol-nitrosoguanidines
- Studies on Cinnolines. II. On Nitration of Cinnoline 1-Oxide
- On Nitration of Cinnoline 1-Oxide
- Reactions of 1-Nitroso-1-phenyl-3-(4-pyridylmethyl)ureas
- Cyclization of (2-Hydroxyethyl) urea Derivatives to Give 3-Nitroso-2-oxazolidinones under Usual Nitrosation Conditions
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- Nitrosation of 1,3-Diarylureas with Nitrosyl Chloride, Dinitrogen Trioxide and Dinitrogen Tetroxide in Dimethylformamide
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- Thermal Decomposition of 1,3-Diaryl-1-nitrosoureas in Benzene
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