Studies on Tertiary Amine Oxides. XXXVIII. Reaction of Quinoline 1-Oxide with N-Acylmethylpyridinium Salts in the Presence of Acylating Agents
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概要
- 論文の詳細を見る
Quinoline 1-oxide (I) was found to react readily with N-acylmethylpyridinium salts (II) in the presence of acetic anhydride to give N-(α-acyl-2-quinolylmethyl) pyridinium salts (III) in good yields, but no reaction was observed without acetic anhydride. Treatment of benzoyl-adduct of quinoline 1-oxide (Ia) with II in the presence of acetic anhydride also afforded III, but the yields of III were somewhat less compared with the former procedure.
- 公益社団法人日本薬学会の論文
- 1970-05-25
著者
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浜名 政和
Faculty of Pharmaceutical Sciences, Kyushu University
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野田 寛治
Research Laboratories Hisamitsu Pharmaceutical Co. Inc.
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浜名 政和
Faculty Of Pharmaceutical Sciences Kyushu University
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山崎 企善
Faculty Of Pharmaceutical Sciences Fukuoka University
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野田 寛治
Faculty of Pharmaceutical Sciences, Fukuoka University
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