Amino Acids and Peptides. XLVII. Facile Synthesis of Flavacol, Deoxymuta-aspergillic Acid and Optically Active Deoxyaspergillic Acid from Dipeptidyl Aldehydes

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概要

• 論文の詳細を見る

• 2(1H)-Pyrazinone ring-containing natural products, flavocol, deoxymuta-aspergillic acid and finally optically active deoxyaspergillic acid, were easily synthesized by a newly developed procedure for preparation of 2(1H)-pyrazinone derivatives from dipeptidyl aldehyde hydrochlorides. The absolute configuration of natural deoxyaspergillic acid was synthetically determined as S.

• 公益社団法人日本薬学会の論文
• 1996-12-15

著者

• Taguchi Hiroyuki

  College Of Pharmacy Nihon University

• OKADA Yoshio

  Faculty of Pharmaceutical Sciences, Kobe Gakuin University

• Okada Yoshio

  Faculty Of Pharmaceutical Sciences Kobe Gakuin University

• YOKOI Toshio

  Faculty of Pharmaceutical Sciences, Kobe Gakuin University

• YOKOI Toshio

  The Graduate School of Food and Medicinal Sciences, Kobe Gakuin University

• TAGUCHI Hiroaki

  Faculty of Pharmaceutical Sciences, Kobe Gakuin University

• Yokoi T

  Kobe‐gakuin Univ. Hyogo Jpn

• Yamamoto T

  R&d Laboratories Nippon Organon K.k.

• Taguchi H

  Kobe Pharmaceutical Univ. Kobe Jpn

• Taguchi Hiroaki

  Faculty Of Pharmaceutical Sciences Kobe-gakuin University

• Yokoi Toshio

  Faculty Of Pharmaceutical Sciences And High-technology Research Center Kobe-gakuin University

• Tsuda Y

  Faculty Of Pharmaceutical Sciences And High Technology Research Center Kobe Gakuin University

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