SYNTHESIS OF ω-TERT-BUTYL ESTERS OF ASPARTIC ACID AND GLUTAMIC ACID VIA B, B-DIFLUOROBOROXAZOLIDONES

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概要

• 論文の詳細を見る

• B, B-Difluoroboroxazolidones (DFBONs) were synthesized for the first time from salts of amino acid and BF_3・Et_2O, and their properties were examined. DFBONs were used in selective preparation of Glu(OBu^t) and Asp(OBu^t) in good yields under catalysis with BF_3・Et_2O and H_3PO_4. Amberlite XAD-2 resin was successfully employed to purify the above amino acid derivatives.

• 公益社団法人日本薬学会の論文
• 1996-11-15

著者

• Li Wei

  Stevens Institute of Technology

• LI Wei

  Department of Hematology, Affiliated Hospital of Academy of Military Medicine Science

• Li Wei

  Faculty Of Pharmaceutical Sciences Toho University

• OKADA Yoshio

  Faculty of Pharmaceutical Sciences, Kobe Gakuin University

• WANG Jidong

  Department of Synchrotron Radiation Science, The Graduate University for Advanced Studies

• Li W

  Faculty Of Pharmaceutical Sciences Toho University

• Okada Yoshio

  Faculty Of Pharmaceutical Sciences Kobe Gakuin University

• WANG Yuanshu

  Institute of Materia Medica, Shandong Academy of Medical Sciences

• Li Wei

  Department Of Molecular Biology Jilin University

• Li W

  Laboratory Of Pharmaceutical Resource Discovery Dalian Institute Of Chemical Physics Chinese Academy

• Wang Yuhong

  Department Of Molecular Biology Jilin University

• Wang Yuhong

  Department Of Anatomy Biology And Medicine Oita University School Of Medicine

• Wang J

  Shenyang Pharmaceutical Univ. Shenyang Chn

• Wang Y

  Institute Of Materia Medica Shandong Academy Of Medical Sciences

• WANG Zongmu

  Department of Molecular Biology, Jilin University

• Wang Zongmu

  Department Of Molecular Biology Jilin University

• Wang Jidong

  Department Of Synchrotron Radiation Science The Graduate University For Advanced Studies

• Wang Jidong

  Department Of Molecular Biology Jilin University

• Wang J

  Department Of Synchrotron Radiation Science The Graduate University For Advanced Studies

• Li Wei

  Department Of Chinese Material Medicine Chinese Material Medicine College Of Jilin Agricultural Univ

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