Synthesis of a New Allosamidin Analog, N,N'-Diacetyl-β-Chitobiosyl Allosamizoline, and Its Inhibitory Activity against Some Chitinases

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概要

• 論文の詳細を見る

• A new allosamidin analog (2), possessing an N,N'-diacetylchitobiosyl moiety as a constituent, was stereoselectively synthesized through the coupling reaction between the disaccharide thioglycoside derivative (5) and allosamizoline derivative (6). The inhibitory activity of 2 against chitinases derived from an insect, yeast and mold were tested and compared with that of allosamidin (1).

• 社団法人日本農芸化学会の論文
• 1993-12-23

著者

• 作田 庄平

  東京大学大学院農学生命科学研究科応用生命化学専攻

• Yamada Yasuhiro

  Department Of Biotechnology Osaka University

• Sakuda S

  Department Of Applied Biological Chemistry The University Of Tokyo

• Yamada Y

  Osaka Univ. Osaka Jpn

• Yamada Y

  Department Of Biotechnology Faculty Of Engineering Osaka University

• SAKUDA Shohei

  Department of Applied Biological Chemistry, University of Tokyo

• KUZUHARA Hiroyoshi

  The Institute of Physical and Chemical Research (RIKEN)

• Sakuda Shohei

  Department Of Applied Biological Chemistry Graduate School Of Agricultural And Life Sciences The Uni

• Takahashi S

  Akita Res. Inst. Food And Brewing Akita

• TAKAHASHI Shunya

  The Institute of Physical and Chemical Research (RIKEN)

• Terayama Hiroyuki

  The Institute of Physical and Chemical Research (RIKEN)

• Terayama Hiroyuki

  Graduate School of Science and Engineering, Saitama University

• 作田 庄平

  東大 大学院

• Kuzuhara H

  Department Of Functional Moterials Science Faculty Of Engineering Saitama University

• Suzuki Takahito

  Biological Laboratory Faculty Of Science Nara Women's University

• Yamada Yasuhiro

  Department Of Agricultural Chemistry Faculty Of Agriculture University Of Tokyo

• SAKUDA Shohei

  Department of Agricultural Chemistry, The University of Tokyo

• Kuzuhara Hiroyoshi

  The Institute of Physical and Chemical Research

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