34 キノールアセタートを経由するイソキノリンアルカロイドの合成
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概要
- 論文の詳細を見る
Pb(OAc)_4 oxidation of 7-hydroxy-6-methoxy-2-methyltetrahydro-isoquinolines possessing electron-donating group at C-3' position in the benzene nucleus of 1-benzyl or 1-phenethyl group, gave the corresponding p-quinol acetates. By the treatment of the p-quinol acetate with various acids, we succeeded in the syntheses of some aporphine, homoaporphine and homomorphinandienone type alkaloids. This cyclization reaction is new, and supplies the useful method for syntheses of some isoquinoline alkaloids.
- 天然有機化合物討論会の論文
- 1973-10-01
著者
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原 博
Faculty Of Pharmaceutical Sciences Science University Of Tokyo
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原 博
東京理科大学薬学部
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大山 恵子
Faculty of Pharmaceutical Sciences, Science University of Tokyo
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利岡 佶
Faculty Of Pharmaceutical Sciences Science University Of Tokyo
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梅澤 文輔
Faculty Of Pharmaceutical Sciences Science University Of Tokyo
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星野 修
東理大薬
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芹沢 信明
Faculty Of Pharmaceutical Sciences Science University Of Tokyo
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星野 修
Faculty Of Pharmaceutical Sciences Science University Of Tokyo
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梅澤 文輔
東理大薬
-
原 博
東理大薬
-
利岡 佶
東理大薬
-
芹沢 信明
東理大薬
-
大山 恵子
東理大薬
-
大山 恵子
Faculty Of Pharmaceutical Sciences Science University Of Tokyo
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