Studies on Tetrahydroisoquinolines. XVII. A Synthesis of 8-Halo-1,2,3,4-tetrahydroisoquinolines
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概要
- 論文の詳細を見る
Treatment with conc. hydrochloric acid of p-quinol acetates (1) obtained from 7-hydroxy-1,2,3,4-tetrahydroisoquinolines (4) gave the corresponding 8-chloro-7-hydroxy-1,2,3,4-tetrahydroisoquinolines (5) in good yields. Similarly, by using conc. hydrobromic acid or 38% hydriodic acid, 8-bromo (6)- or 8-iodo-corypalline (7) was obtained.
- 公益社団法人日本薬学会の論文
- 1981-01-25
著者
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星野 修
東京理科大学薬学部
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原 博
Faculty Of Pharmaceutical Sciences Science University Of Tokyo
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原 博
東京理科大学薬学部
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星野 修
Faculty of Pharmaceutical Sciences, Science University of Tokyo
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梅澤 文輔
Faculty of Pharmaceutical Sciences, Science University of Tokyo
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梅澤 文輔
Faculty Of Pharmaceutical Sciences Science University Of Tokyo
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原 博
東京理大 薬
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星野 修
Faculty Of Pharmaceutical Sciences Science University Of Tokyo
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