Electrophilic Substitution of 1,2-Benzisothiazol-3-acetic Acid
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概要
- 論文の詳細を見る
The bromination, the nitration, the chlorosulfonation, the formylation and the Mannich reaction of 1,2-benzisothiaizol-3-acetic acid (1) were investigated and it was shown that the 3α-methylene group is also activated to the electrophilic substitutions as in 1,2-benzisoxazol-3-acetic acid.
- 公益社団法人日本薬学会の論文
- 1978-12-25
著者
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宇野 準
大日本製薬株式会社総合研究所
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黒川 美貴雄
Research Laboratories, Dainippon Pharmaceutical Co., Ltd.
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宇野 準
大日本製薬株式会社
-
宇野 準
大日本製薬
-
宇野 準
Research Laboratory Dainippon Pharmaceutical Co. Ltd.
-
黒川 美貴雄
大日本製薬株式会社創薬研究所
-
宇野 準
Research Laboratories Dainippon Pharmaceutical Co. Ltd.
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