Synthesis of p-Boronophenylserine, a New Boron-containing Amino Acid for Boron Neutron Capture Therapy
スポンサーリンク
概要
- 論文の詳細を見る
The synthesis of p-boronophenylserine (BPS), a new water-soluble analogue of p-boronophenylalanine (BPA), was achieved from p-[(dihydroxy)boryl] benzaldehyde (1) in four steps. The key intermediate, oxazoline(4), was prepared by the reaction of the protected aldehyde(2) with ethyl isocyanoacetate(3), using sodium cyanide, and then transformed into syn- and anti-BPS.
- 社団法人日本農芸化学会の論文
- 1995-12-23
著者
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KIRIHATA Mitsunori
Department of Agriculture, Osaka Prefectural University
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Miyatake K
Osaka Prefecture Univ. Osaka Jpn
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ICHIMOTO Itsuo
Department of Agricultural Chemistry, Faculty of Agriculture, University of Osaka Prefecture
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MATSUDA Kazuhiko
Laboratory of Plant Pathology and Biotechnology and Laboratory of Pesticide Chemistry
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切畑 光統
大阪府立大学 農学部
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Kirihata Mitsunori
Graduate School Of Life And Environmental Science Osaka Prefecture University
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Kirihata Mitsunori
Department Of Agricultural Chemistry College Of Agriculture University Of Osaka Prefecture
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Ichimoto I
Department Of Applied Biochemistry College Of Agriculture University Of Osaka Prefecture
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Ichimoto Itsuo
Department Of Agricultural Chemistry College Of Agriculture
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Morimoto T
Department Of Applied Biological Chemistry The University Of Tokyo
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MORIMOTO Tsuguhiro
Department of Applied Biochemistry, College of Agriculture, University of Osaka Prefecture
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Mizuta Takanori
Department of Applied Biochemistry, College of Agriculture, University of Osaka Prefecture
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Morimoto T
Kagawa Univ. Kagawa Jpn
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Morimoto Tsuguhiro
Department Of Applied Biochemistry College Of Agriculture University Of Osaka Prefecture
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Mizuta Takanori
Department Of Applied Biochemistry College Of Agriculture University Of Osaka Prefecture
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KIRIHATA Mitsunori
Department of Agricultual Chemistry, College of Agriculture, University of Osaka Prefecture
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