Synthesis and Biological Evaluation of Peptide Mimics Derived from First Extracellular Loop of CCR5 toward HIV-1
スポンサーリンク
概要
- 論文の詳細を見る
Peptide mimics derived from the first extracellular loop of CCR5 bearing non-peptide spacers in place of Ala-Ala-Ala sequence in the peptide moiety were synthesized, and the effects of these compounds on the inhibition against HIV-1 were examined. Compound 2b having m-aminophenoxyacetic acid derivative as a non-peptide spacer significantly inhibited HIV-1.
- 公益社団法人日本薬学会の論文
- 2004-12-01
著者
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池田 潔
School Of Pharmaceutical Sciences University Of Shizuoka
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Konishi K
School Of Pharmaceutical Sciences University Of Shizuoka
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Tanaka K
Department Of Molecular Engineering Graduate School Of Engineering Kyoto University
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池田 潔
Tanabe Seiyaku Co. Ltd. Saitama Jpn
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Ishii Y
School Of Pharmaceutical Sciences University Of Shizuoka
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Tanaka Ken-ichiro
Faculty Of Pharmaceutical Sciences Okayama University
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TANAKA Kiyoshi
School of Pharmaceutical Sciences, University of Shizuoka
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IKEDA Kiyoshi
School of Pharmaceutical Sciences, University of Shizuoka
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ISHII Yuko
School of Pharmaceutical Sciences, University of Shizuoka
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KONISHI Koji
School of Pharmaceutical Sciences, University of Shizuoka
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SATO Masayuki
School of Pharmaceutical Sciences, University of Shizuoka
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Tanaka Katsuyuki
Dept. Biol. Sci. Fac. Sci. Hiroshima Univ.
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Ikeda Kiyoshi
Department Of Biochemistry Osaka University Of Pharmaceutical Sciences
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Tanaka K
Dept. Biol. Sci. Fac. Sci. Hiroshima Univ.
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池田 かおり
Developmental Research Laboratories Shionogi & Co. Ltd.
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Ikeda Kaori
Developmental Research Laboratories Shionogi & Co. Ltd.
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Ishii Yuko
School Of Pharmaceutical Sciences University Of Shizuoka
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Tanaka Kiyoshi
School Of Pharmaceutical Sciences University Of Shizuoka
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Konishi K
Nippon Dental Univ. Tokyo Jpn
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Ikeda Kiyoshi
School Of Information Science Japan Advanced Institute Of Science And
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Sato Masayuki
School Of Pharmaceutical Sciences University Of Shizuoka
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Sato Masayuki
School Of Pharmaceutical Sciences Univ. Of Shizuoka
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