Studies on Thioamides. II. Application of Thioamides in Bischler-Napieralski Reaction.

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概要

• 論文の詳細を見る

• Thioamides have been cyclized in good yield to the corresponding 1-substituted 3,4-dihydroisoquinoline under the normal Bischler-Napieralski reaction conditions which are generally used to cyclize acid amides. Phosphorus pentasulfide has been effectively used as a condensing agent in the Bischler-Napieralski reaction to get 1-substituted-3,4-dihydroquinoline from both thioamides as well as normal acid amides.

• 公益社団法人日本薬学会の論文
• 1964-02-25

著者

• 山田 俊一

  Faculty of Pharmaceutical Sciences, University of Tokyo

• アブドールーモハッセン エム.イー.オマール

  Faculty of Pharmaceutical Sciences, University of Tokyo

• 山田 俊一

  Faculty Of Pharmaceutical Sciences University Of Tokyo

• アブドールーモハッセン エム.イー.オマール

  Faculty Of Pharmaceutical Sciences University Of Tokyo

関連論文

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