Reaction of 3-Formylrifamycin SV with Formalin in Combination with Primary Alkylamines
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概要
- 論文の詳細を見る
3-Formylrifamycin SV (4) was found to react with formalin in combination with primary alkylamines to give 2,3-dihydropyrimido [4,5-b] rifamycin derivatives 3. The iminium carbon of 3 was found to be reduced when primary alkylamines with at least one hydrogen atom at the α-position were used. The addition of an alcoholic OH group to the iminium carbon of 3 is also described.
- 公益社団法人日本薬学会の論文
- 1980-08-25
著者
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塚本 悟郎
Pharmaceuticals Research Center, Kanebo Ltd.
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塚本 悟郎
New Drug Research Laboratories Kanebo Ltd.
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相川 法男
Pharmaceuticals Research Center, Kanebo, Ltd.
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田口 雅裕
Pharmaceuticals Research Center Kanebo Co. Ltd.
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相川 法男
Pharmaceuticals Research Center
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塚本 悟郎
Pharmaceutical Research Laboratory, Tanabe Seiyaku Co., Ltd.
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