Studies on the Syntheses of Heterocyclic Compounds. DCCLXVIII. Reaction of Pyrrolo [1,2-a] indole Derivatives with N-Bromosuccinimide in Protic Solvents
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概要
- 論文の詳細を見る
Treatment of the 2,3-dihydro-1H-pyrrolo [1,2-a] indoles (1 and 7) with N-bromosuccinimide in protic solvents such as methanol and acetic acid yielded the brominated compounds (4 and 8). The reaction of the pyrrolo [1,2-a] indole-5,8-diones (9-13) with N-bromosuccinimide in these solvents afforded the adducts (14-18 and 20-21). Debromination of the brominated compounds (5b, 15,16 and 20) with tri-n-butyltin hydride was also described.
- 社団法人日本薬学会の論文
- 1978-12-25
著者
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井原 正隆
東北大院薬
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亀谷 哲治
Pharmaceutical Institute, Tohoku University School of Medicine
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福本 圭一郎
東北大・薬
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福本 圭一郎
Pharmaceutical Institute, Tohoku University
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高橋 喜美男
Pharmaceutical Institute, Tohoku University
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井原 正隆
Pharmaceutical Institute, Tohoku University
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井原 正隆
東北大薬
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井原 正隆
東北大学薬学部
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亀谷 哲治
Pharmaceutical Institute Medical Faculty University Of Osaka
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福本 圭一郎
Pharmaceutical Institute Tohoku University School Of Medicine
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高橋 喜美男
Pharmaceutical Institute Tohoku University
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