Nitrenes. VIII. A Novel Synthesis of 3-Cyano-2-ethoxy-6,7-disubstitutedquinolines with Triethyl Phosphite (Studies on the Syntheses of Heterocyclic Compounds. CDXVI)

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概要

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• Treatment of ethyl 3,4-disubstituted-benzylidenecyanoacetate (V, VI and VII), whose ethoxycarbonyl group was oriented in the trans configuration to the benzene ring, with triethyl phosphite afforded the 3-cyano-2-ethoxy-6,7-disubstituted-quinolines (XI, XII, and XIII) in good yield.

• 公益社団法人日本薬学会の論文
• 1971-07-25

著者

• 亀谷 哲治

  Pharmaceutical Institute, Tohoku University School of Medicine

• 山中 徹

  東北大・薬

• 丹生 淳郷

  Pharmaceutical Institute, Tohoku University

• 山中 徹

  Pharmaceutical Institute, Tohoku University

• 亀谷 哲治

  Pharmaceutical Institute Medical Faculty University Of Osaka

• 丹生 淳郷

  日本ケミファ株式会社研究部

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