Studies of Heterocyclic Compounds. XVII. Synthesis of 3-(Substituted-phenyl)-thiazolo [2,3-b] benzothiazolium Perchlorates

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概要

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• Seventeen 3-(substituted-phenyl) thiazolo [2,3-b] benzothiazolium perchlorates (3) were synthesized by acid-cyclization of the ketosulfides (2), which were prepared by alkylation of 2-mercaptobenzothiazole sodium salt with substituted phenacyl halides (1). Some of the phenacyl halides were prepared by chloroacetylation of substituted benzenes, and the others by bromination of the corresponding substituted acetophenones.

• 公益社団法人日本薬学会の論文
• 1977-12-25

著者

• 宮坂 貞

  School of Pharmaceutical Sciences, Showa University

• 澤田 誠吾

  Yakult Central Institute of Microbiological Research

• 澤田 誠吾

  ヤクルト本社中央研究所

• Sawada S

  Yakult Central Institute Of Microbiological Research

• 宮坂 貞

  School Of Pharmaceutical Sciences Showa University

• 沢田 誠吾

  School of Pharmaceutical Sciences, Showa University

• 荒川 基一

  School of Pharmaceutical Sciences, Showa University

• 荒川 基一

  School Of Pharmaceutical Sciences Showa University

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