A NOVEL AND REGIOSPECIFIC ROUTE TO 5-ACYLURIDINES VIA AN AMIDE α-ANION DERIVED FROM 5,6-DIHYDROURIDINE
スポンサーリンク
概要
- 論文の詳細を見る
Upon lithiation with LDA, 2', 3'-O-isopropylidene-5'-O-methoxymethyl-5,6-dihydrouridine has been shown to serve as an "amide α-anion". Thus, acylation of the resulting dianion took place regiospecifically at the C-5 position. The subsequent phenylselenenylation and oxidative elimination afforded 5-acyluridines.
- 公益社団法人日本薬学会の論文
- 1982-12-25
著者
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田中 博道
School of Pharmaceutical Sciences, Showa University
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宮坂 貞
School of Pharmaceutical Sciences, Showa University
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宮坂 貞
昭和大学大学院薬学研究科医療薬学専攻
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早川 弘之
School of Pharmaceutical Sciences, Showa University
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宮坂 貞
School Of Pharmaceutical Sciences Showa University
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