Short-step Syntheses of All Stereoisomers of Preussin and Their Bioactivities(Organic Chemistry)
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概要
- 論文の詳細を見る
All the eight stereoisomers of (+)-preussin (1b), an antifungal agent inhibiting the growth of fission yeast and human cancer cells, were synthesized in two steps by non-stereoselective reactions and chromatographic separation, starting from L- and D-N-protected-phenylalaninal (2). Their bioassay revealed all of the stereoisomers to be almost equally bioactive.
- 社団法人日本農芸化学会の論文
- 2002-05-23
著者
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Yoshida Minoru
Department of Thoracic and Cardiovascular Surgery, Wakayama Medical University School of Medicine
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Kitahara Takeshi
Department Of Applied Biological Chemistry Division Of Agriculture And Agricultural Life Science The
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HORINOUCHI Sueharu
Department of Biotechnology, University of Tokyo
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WATANABE HIDENORI
Department of Applied Biological Chemistry, The University of Tokyo
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Yoshida M
Department Of Biotechnology Graduate School Of Agricultural And Life Sciences The University Of Toky
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OKUE Masayuki
Department of Applied Biological Chemistry, Graduate School of Agricultural and Life Sciences, The U
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KASAHARA Koji
Science and Biological Supramolecular Systems, Graduate School of Integrated Science, Yokohama City
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Horinouchi Sueharu
Department Of Biotechnology Graduate School Of Agricultural And Life Sciences The University Of Toky
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Horinouchi Sueharu
Department Of Agricultural Chemistry Faculty Of Agriculture University Of Tokyo
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Horinouchi Sueharu
Department Of Agricultural Chemistry Faculty Of Agriculture The University Of Tokyo
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Horinouchi Sueharu
Dep. Of Biotechnology Graduate School Of Agriculture And Life Sciences Univ. Of Tokyo
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Okue Masayuki
Department Of Applied Biological Chemistry Graduate School Of Agricultural And Life Sciences The Uni
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Kasahara Koji
Science And Biological Supramolecular Systems Graduate School Of Integrated Science Yokohama City Un
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Watanabe H
The University Of Tokyo
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Kitahara T
The University Of Tokyo
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Kitahara T
Department Of Agricultural Chemistry The University Of Tokyo
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Horinouchi S
Department Of Biotechnology The University Of Tokyo
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Watanabe Hidenori
Department Of Applied Biological Chemistry Graduate School Of Agricultural And Life Sciences The Uni
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Watanabe Hidenori
Department Of Applied Biological Chemistry Graduate School Of Agricultural And Life Sciences The Uni
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Kitahara Takeshi
Department Of Agricultural Chemistry The University Of Tokyo
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Kitahara Takeshi
Department Of Applied Biological Chemistry Graduate School Of Agricultural And Life Sciences The Uni
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Watanabe Hidenori
Department Of Applied Biological Chemistry Graduate School Of Agricultural And Biological Sciences T
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Yoshida Minoru
Department Of Chemistry St. Marianna University School Of Medicine
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Yoshida Minoru
Department Of Agricultural Chemistry Faculty Of Agriculture Iwate University
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Kitahara Takeshi
School Of Pharmacy Teikyo Heisei Univ.
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