Insecticidal and Antifungal Activities of Aminorhodanine Derivatives

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概要

• 論文の詳細を見る

• Aminorhodanine (1) showed strong insecticidal activity against Culex pipiens pallens and Musca domestica, with respective LD_<50> values of 0.21μg/insect and 0.87μg/insect. Compound 1 had antifungal activity against Aspergillus niger ATCC-16404,Trichophyton mentagrophytes IFO-32412,Candida albicans ATCC-10231,Hansenula anomala OPS-308 and Penicillium expansum IFO-8800. In particular, 1 had potent antifungal activity against Aspergillus niger ATCC-16404,its minimal inhibitory concentration (MIC) being 6.25μg/ml. Both activities of 1 were much higher than those of rhodanine (4), suggesting that the introduction of an amino group into N-3 of 4 plays an important role in the biological activity of rhodanine-related compounds. On the other hand, N-acetylaminorhodanine (2) and N-benzoylaminorhodanine (3) did not show either activity, suggesting that the free amino group at N-3 of 1 is closely related to the inhibitory activity of rhodanine derivatives.

• 社団法人日本農芸化学会の論文
• 1998-05-23

著者

• NUMATA Atsushi

  Graduate School of Pharmaceutical Sciences, Tohoku University

• TSUJIBO Hiroshi

  Osaka University of Pharmaceutical Sciences

• INAMORI Yoshihiko

  Osaka University of Pharmaceutical Sciences

• NUMATA Atsushi

  Osaka University of Pharmaceutical Sciences

• SAKAGAMI YOSHIKAZU

  Osaka Prefectural Institute of Public Health

• SAKAGAMI YOSHIKAZU

  Kinki University, Faculty of Agriculture

• SHIBATA Mitsunobu

  Fumakilla Ltd.

• KUMEDA Yuko

  Osaka Prefectural Institute of Public Health

• Sakagami Yoshikazu

  Kinki University Faculty Of Agriculture

• Sakagami Y

  Osaka Prefectural Institute Of Public Health

• Takegawa Yoko

  Osaka University Of Pharmaceutical Sciences

• OKAMOTO Yukiko

  Osaka University of Pharmaceutical Sciences

• Okamoto Yukiko

  Laboratory Of Food Biochemistry Division Of Applied Bioscience Graduate School Of Agriculture Hokkai

• Numata A

  Graduate School Of Pharmaceutical Sciences Tohoku University

• Numata A

  Osaka University Of Pharmaceutical Sciences

• Numata Atsushi

  Osaka College Of Pharmacy

• Numata Atsushi

  Osaka Univ. Pharmaceutical Sci. Osaka Jpn

• Inamori Yoshihiko

  Osaka College Of Pharmacy

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