NEW METHODS AND REAGENTS IN ORGANIC SYNTHESIS. 44. A NEW GENERAL EFFICIENT SYNTHESIS OF DL-[N]-GINGEROLS AND RELATIVES THROUGH DIRECT C-ACYLATION USING DIETHYL PHOSPHOROCYANIDATE (DEPC)

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概要

• 論文の詳細を見る

• DL-[n]-Gingerols (1) and their relatives, which have various interesting physiological actions, have been conveniently and efficiently prepared from ferulic acid (2) through direct C-acylation using diethyl phosphorocyanidate (DEPC) in the presence of triethylamine.

• 1984-04-25

著者

• 浜田 康正

  Faculty of Pharmaceutical Sciences, Nagoya City University

• 塩入 孝之

  Faculty of Pharmaceutical Sciences, Nagoya City University

• 加藤 信治

  Central Research Laboratories, Santen Pharmaceutical Co., Ltd.,

• 塩入 孝之

  Faculty Of Pharmaceutical Sciences Nagoya City University

• 塩入 孝之

  名古屋市大・薬

• 加藤 信治

  Central Research Laboratories Santen Pharmaceutical Co. Ltd.

• 加藤 信治

  Faculty of Pharmaceutical Sciences, Nagoya City University

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