A CONVENIENT METHOD FOR THE SYNTHESIS OF αβ-UNSATURATED CARBOXYLIC ACID AMIDES UTILIZING A NEW HETERO-BIFUNCTIONAL REAGENT, DMPATT

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概要

• 論文の詳細を見る

• As a new extention of monitored aminolysis of 3-acyl-1,3-thiazolidine-2-thione (ATT), a convenient procedure for the synthesis of αβ-unsaturated carboxylic acid amides has been developed using a new hetero-bifunctional reagent, 3-dimethylphosphonoacetyl-1,3-thiazolidine-2-thione (DMPATT). DMPATT was effectively used as the bridging reagent between amino (or imino) compounds and aldehydes (or ketone) to afford various olefinic amides in good yields.

• 公益社団法人日本薬学会の論文
• 1984-11-25

著者

• 藤田 榮一

  Osaka University of Pharmaceutical Sciences

• 長尾 善光

  Institute for Chemical Research, Kyoto University

• 落合 正仁

  Institute for Chemical Research, Kyoto University

• 山田 省三

  Institute For Chemical Research Kyoto University

• 藤田 榮一

  Institute for Chemical Research, Kyoto University

• 長尾 善光

  Institute For Chemical Research Kyoto University

• 萩原 裕一

  Institute for Chemical Research, Kyoto University

• 萩原 裕一

  京都大学化学研究所

• 落合 正仁

  Institute For Chemical Research Kyoto University

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