PROPERTIES OF N^α, N^<ca>-DI- TERT-BUTYLOXYCARBONYL-ω-CARBAMOYL-α-AMINO ACIDS AND DIRECT SYNTHESIS OF PROTECTED HOMOGLUTAMIC ACID DERIVATIVES
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概要
- 論文の詳細を見る
The protected carboxamide function of N^α, N^<ca>-di-tert-butyloxycarbonyl-ω-carbamoyl-α-amino acids worked well with nucleophilic reagents. Applying this novel reactivity, we developed an efficient synthetic route to N^α-tert-butyloxycarbonylhomoglutamic acid and its derivatives, including N^α-tert-butyloxycarbonylhomoglutamic acid δ-benzyl ester, from N^α, N^<ca>-di-tert-butyloxycarbonylhomoglutamine.
- 社団法人日本薬学会の論文
- 1986-08-25
著者
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広瀬 恭子
Faculty of Pharmaceutical Sciences, Hokuriku University
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橋本 忠
北陸大・薬
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佐倉 直樹
北陸大・薬
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Sakura Naoki
Faculty Of Pharmaceutical Sciences Hokuriku University
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佐倉 直樹
School of Pharmacy, Hokuriku University
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橋本 忠
School of Pharmacy, Hokuriku University
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広瀬 恭子
School of Pharmacy, Hokuriku University
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Hashimoto T
Hokuriku Univ. Kanazawa Jpn
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Hashimoto Toshihiro
Fac. Of Pharmaceutical Sciences Tokushima Bunri Univ.
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広瀬 恭子
Faculty Of Pharmaceutical Sciences Hokuriku University
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橋本 忠
School Of Pharmacy Tokyo University Of Pharmacy And Life Sciences
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