Studies of Alicyclic α-Amino Acids. III. Synthesis and Biological Evaluation of 3-Amino-1,2,3,4-tetrahydrocarbazole-3-carboxylic Acids
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概要
- 論文の詳細を見る
3-Amino-1,2,3,4-tetrahydrocarbazole-3-carboxylic acid (IIa) and its 6-methoxy, benzyloxy and hydroxy derivatives (IIb-d), a new type of cyclic tryptophan analogue, were prepared. The optical resolution of acetamido-(-)-menthyl ester of IIa (XIIc) was achieved. It was found that IIa inhibited α-chymotrypsin competitively and trypsin noncompetitively.
- 公益社団法人日本薬学会の論文
- 1973-11-25
著者
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小木曾 太郎
Faculty of Pharmaceutical Sciences, Kinki University
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牧 敬文
Gifu College Of Pharmacy
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小木曾 太郎
Gifu College Of Pharmacy
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小木曾 太郎
Faculty Of Pharmaceutical Sciences Kinki University
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平光 時幸
Gifu College of Pharmacy
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馬杉 峻
Gifu College of Pharmacy
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