Isocarbostyril関連化合物の合成研究(第3報)2-Methyl-3-aminoisocarbostyrilとp-置換ベンズアルデヒドの反応
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概要
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Reaction of 3-aminio-2-methylisocarbostyril with an aromatic aldehyde generally gave the corresponding Schiff base and the corresponding novel pyrido[2,3-c ; 6,5-c']diisoquinoline-5,9-dione derivatives. In order to examine the generality of this reaction, the reaction was carried out under various conditions using several aromatic aldehydes having electron-releasing or electron-attracting substituents (-CH_3,-OCH_3,-Cl, -NO_2) in the para-position. The reaction mechanism was presented from these results.
- 公益社団法人日本薬学会の論文
- 1972-12-25
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