Isocarbostyril 関連化合物の合成研究(第1報) : 2-Methyl-3-aminoisocarbostyril と酸クロリドの反応
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Reactions of 2-methyl-3-aminoisocarbostyril (I) with several acid anhydrides and acid chlorides were examined using acetic anhydride, acetyl chloride, benzoic anhydride, benzoyl chloride, oxalyl chloride and trans-cinnamoyl chloride. Acylation of C-4 in I, giving II, V, and X, took place predominantly in these cases, although the reaction of I with acryloyl chloride gave VIIa as the main product.
- 公益社団法人日本薬学会の論文
- 1971-12-25
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