Isocarbostyril関連化合物の合成研究(第6報) 3-Alkoxyisocarbostyril誘導体の合成と反応
スポンサーリンク
概要
- 論文の詳細を見る
3-Alkoxyisocarbostyrils (IIa-e) were synthesized from 2-cyanomethylbenzoate (I) by heating with various primary alcohols in the presence of an equivalent amount of sodium. It was found that 3-methoxyisocarbostyril (IIa) reacted easily with hydrazine hydrate and mono- or di-substituted amines to give the corresponding 3-substituted aminoisocarbostyrils (VIIIa-i) in a good yield.
- 公益社団法人日本薬学会の論文
- 1976-02-25
著者
関連論文
- Studies on Synthesis and Stereochemistry of 3-Methyloctahydroisocoumarins and 1-Methyloctahydro-3H-2-benzopyran-3-ones
- Studies on Synthesis of 10,11-Dihydro-5H-dibenzo[a, d]cycloheptene Derivatives. IV. : Photoreactions of 5-Substituted-5H-dibenzo[a, d]cycloheptenes with 1,2-Substituted Olefins and the Stereostructures of the Cycloaddition Products
- Studies on Synthesis of 10,11-Dihydro-5H-dibenzo[a, d]cycloheptene Derivatives, III. : Stereostructures of Isomeric 8,9-Dimethoxycarbonyldibenzo[2,3 : 5,6]bicyclo[5.2.0]nonan-4-ones Determined by ^1H-^1H and ^C-{^1H}Nuclear Overhauser Effects in Nucle
- Synthesis and Application of Imidazole Derivatives. Synthesis of 5-Methyl-7,8,9,10-tetrahydro-5H-azepino[1,2-α]benzimidazol-7-one and Related Compounds
- A Total Synthesis of Grifolin
- Synthesis and Application of Imidazole Derivatives : Preparation of Various Diketones from 1,n-Bis(1-methyl-1H-imidazol-2-yl)alkane-1,n-diones
- Synthesis and Application of Imidazole Derivatives. : Synthesis of (1-Methyl-1H-imidazol-2-yl)methanol Derivatives and Conversion into Carbonyl Compounds(Organic,Chemical)
- An Efficient Biogenetic-Type Transformation of 3-Tertiary-hydroxyalkanoic Acids to Olefinic Compounds(Organic,Chemical)
- Synthesis and Application of Imidazole Derivatives. Synthesis and Acyl Activation of 2-Acyl-1-methyl-1H-imidazoles(Organic,Chemical)
- 2-Amino-1,2,3,4-tetrahydroisoquinoline-1,3-dione並びにその誘導体の抗炎症, 鎮痛及び解熱作用
- tert-Butyl Carboxylatesの一改良合成法について
- 合成化学における1-Acylimidazoleの新しい利用
- 縮合Indole-4,7-dione関連化合物の合成研究(第3報)γ-Amino-n-butyric Acidおよびγ-Amino-β-hydroxy-n-butyric Acidを用いるPyrrole-2-acetic Acid誘導体の合成
- Use of β-Ketocarboxylic Acids for Syntheses of 6-Substituted 4-Hydroxy-2-pyrones and Acyclic β-Diketones
- 10,11-Dihydro-5H-dibenzo[a, d]cycloheptene誘導体の合成研究
- A Novel and Versatile Separation Method for Aldehydes
- Studies on the Syntheses of Condensed Indole-4,7-diones. II. Synthesis of Pyrrolo [1,2-a] indole-5,8-dione Derivatives
- 縮合Indole-4,7-dione関連化合物の合成研究(第1報)2,3-Dichloronaphthoquinoneを出発原料とするBenz[f]indole-4,9-dione誘導体の合成
- デカハイドロイソキノリン誘導体の立体化学(第12報) 2-Methyl-7-amino-cis-decahydroisoquinolineの合成
- Isocarbostyril関連化合物の合成研究(第7報) 2-MethylhomophthalimideとCH_2N_2の異常反応
- Isocarbostyril関連化合物の合成研究(第6報) 3-Alkoxyisocarbostyril誘導体の合成と反応
- Stereochemistry of 3-Methylhexahydrophthalide
- Isocarbostyril関連化合物の合成研究(第5報)2-Acylamido-3-aminoisocarbostyrilの閉環反応
- Studies on Peptides XVIII. Catalytic Hydrogenation of Methionine-containing Peptides
- The Use of Boron Trifluoride Etherate for Debenzyloxycarbonylation of Methionine-containing Peptides by Catalytic Hydrogenolysis
- デカハイドロイソキノリン誘導体の立体化学(第9報) : cis-4-Hydroxy-2-methyldecahydroisoquinolineの合成
- Stereochemistry of Decahydroisoquinolines and Related Compounds. VIII. Syntheses of trans-4-Hydroxy-2-methyldecahydroisoquinolines
- Isocarbostyril関連化合物の合成研究(第4報)2,3-Diaminoisocarbostyrilのアシル化
- デカハイドロイソキノリン誘導体の立体化学(第11報)
- Stereochemistry of 3-Methylhexahydrophthalide
- Isocarbostyril関連化合物の合成研究(第3報)2-Methyl-3-aminoisocarbostyrilとp-置換ベンズアルデヒドの反応
- Isocarbostyril関連化合物の合成研究(第2報)2-Methyl-3-aminoisocarbostyrilとベンズアルデヒドの反応
- Stereochemistry of Decahydroisoquinolines and Related Compounds. X. Configurational Assignment of Epimeric 4-Hydroxy-2-methyl-cis-decahydroisoquinolines
- Isocarbostyril 関連化合物の合成研究(第1報) : 2-Methyl-3-aminoisocarbostyril と酸クロリドの反応
- Stereochemistry of Decahydroisoquinolines and Related Compounds. VII. Syntheses of trans-2-Methyl-1,2,3,4,4a, 5,6,7,8,8a-decahydro-7-isoquinolinols
- 10,11-Dihydrodibenzo[b, f]thiepin誘導体の合成研究
- Studies on Synthesis of 10,11-Dihydro-5H-dibenzo[a, d]cycloheptene Derivatives. II. : Synthesis and Structural Confirmation of Photocycloadducts, 8,9-Dimethoxycarbonyl-2 : 3,5 : 6-dibenzobicyclo[5.2.0] nonan-4-one and Related Compounds : Using Two-Dimensi
- Stereochemistry of Decahydroisoquinolines and Related Compounds. V. Syntheses of 2-Methyl-decahydro-8-isoquinolinols
- Stereochemistry of Decahydroisoquinolines and Related Compounds. III. Syntheses of cis-2-Methyl-decahydro-7-isoquinolinols.
- 10,11-Dihydro-5H-dibenzo[a, d]-cycloheptene誘導体の合成研究
- 合成化学における1-Acylimidazoleの新しい利用
- Studies on the Alkaloids of Amsonia elliptica ROEM ET SCHULT. IV. 17-Ketoyohimbine.
- On the Syntheses of 2-Methyl-7-decahydroisoquinolinols starting from Diethyl 4-Hydroxyhexahydrohomophthalate and Their Configurational Analysis on Their Structure