Introduction of Carbogenic Substituent into the 4-Position of 1-Methyl-1H-imidazole

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概要

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• The 4-position of the 1-methyl-1H-imidazole ring was lithiated by treatment of the corresponding 4-bromo derivatives with tert-butyllithium. This procedure was applied to synthesis of the left-hand part of pyronaamidine (1), which is a biologically interesting marine alkaloid.

• 公益社団法人日本薬学会の論文
• 1994-04-15

著者

• 山本 徹也

  Kyoto Pharmaceutical University

• 太田 俊作

  Kyoto Pharmaceutical University

• 山下 正行

  Kyoto Pharmaceutical University

• 川崎 郁勇

  Kyoto Pharmaceutical University

• 吉川 智子

  Kyoto Pharmaceutical University

• 川崎 郁勇

  京都薬大

• 太田 俊作

  京都薬科大学薬学部

• 長嶋 雄一

  Kyoto Pharmaceutical University

• 太田 俊作

  Kyoto College Of Pharmacy

• 山下 正行

  京都薬科大学薬学部

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