Studies on Steroids. II. The Preparation and Properties of 17β-(N-Substituted 2-Amino-4-thiazolyl) androst-4-en-3β, 17α-diol Series and its Hydrogen Succinate.
スポンサーリンク
概要
- 論文の詳細を見る
17β-(2-alkylamino-(or 2-arylamino-or 2-N, N-alkylarylamino-) thiazolyl) androst-4-en-3β, 17α-diol was prepared from corresponding 3-one with sodium boronhydride in dioxan or dioxane-methanol (1 : 1). 17β-(2-alkylamino-(or 2-arylamino-)-4-thiazolyl) androst-4-en-3β, 17α-diol 3-(hydrogen succinate) and O, N-bis(hydrogen succinate) were obtained from corresponding 3β, 17α-diol and 17α-ol-3-one with succinic anhydride. Some of this substance had a digitalis like properties.
- 社団法人日本薬学会の論文
- 1963-05-25
著者
-
高村 圭一
中外製薬株式会社綜合研究所
-
磯野 千冬
中外製薬綜研
-
磯野 千冬
中外製薬株式会社綜合研究所
-
高村 圭一
Research Laboratory, Chugai Pharmaceutical Co., Ltd.
-
磯野 千冬
Research Laboratory, Chugai Pharmaceutical Co., Ltd.
-
高間 伸一
Research Laboratory, Chugai Pharmaceutical Co., Ltd.
-
新田 義博
Research Laboratory, Chugai Pharmaceutical Co., Ltd.
-
高間 伸一
Research Laboratories Chugai Pharmaceutical Co. Ltd.
-
新田 義博
School Of Pharmacy Hokuriku University
関連論文
- Reaction of Thio Acid S-Esters with p-Toluenesulfonic Acid : A Facile Gynthesis of p-Toluenethiosulfonic S-Esters
- Reaction of Phosphorus Oxyacid Esters with p-Toluenesulfonic Acid
- 101 Chlorpromazine経口投与による偽妊娠誘起について(生理学・薬理学分科会)(第72回日本獣医学会記事)
- 各種系統マウスの化骨時期の比較検討
- スルホンアミド類の合成研究(第3報)1,2,4-Benzothiadiazine 1,1-Dioxide類の合成
- Studies on Steroids. II. The Preparation and Properties of 17β-(N-Substituted 2-Amino-4-thiazolyl) androst-4-en-3β, 17α-diol Series and its Hydrogen Succinate.
- Studies on Steroids. I. The Preparation and Properties of 17β-(N-Substituted 2-Amino-4-thiazolyl)-androst-4-en-3-one Series.
- A New Method for the Synthesis of Amides from Amines : Ruthenium Tetroxide Oxidation of N-Protected Alkylamines
- Chemical Conversion of L-α,ω-Diamino Acids to L-ω-Carbamoyl-α-amino Acids by Ruthenium Tetroxide Oxidation(Organic,Chemical)
- Ruthenium Tetroxide Oxidation of N-Acylated Alkylamines: A New General Syuthesis of Imides(Organic,Chemical)
- A New Approach for the Total Synthesis of L-γ-Carboxyglutamic Acid : Utility of Ruthenium Tetroxide Oxidation
- A Novel Synthesis of L-Pyroglutamic Acid Derivatives from L-Proline : Utility of N-Protecting Groups for Ruthenium Tetroxide Oxidation of Cyclic α-Amino Acids
- Chemical Conversion of Cyclic α-Amino Acids to α-Aminodicarboxylic Acids by Improved Ruthenium Tetroxide Oxidation
- A NOVEL SYNTHESIS OF L-ω-CARBAMOYL-α-AMINO ACIDS FROM L-α, ω-DIAMINO ACIDS BY RUTHENIUM TETROXIDE OXIDATION METHOD
- Pyrimidine Derivatives. III. The Preparation and Bacteriostatic Activity of Benzamidopyrimidines
- Pyridazine Derivatives. X. 10H-Benzo[b]pyridazino[3,4-e][1,4]thiazine and 5H-Benao[b]pyridazino[4,3-e][1,4]thiazine
- Pyridazine Derivatives. VII. Syntheses of 1,2- and 2,3-Diazaphenothiazines
- Kessoglycol 8-Monoacetateの薬理作用
- Kessoglycol誘導体の合成とスクリーニング
- ヤツデのサポニンの研究
- 生薬ならびに植物成分の薬理学的研究(第1報)日本産吉草根の薬理作用
- 2-Substituted Phenethyl-3-[(N, N-dialkyl, or N-cycloalkyl)aminocarbonylethyl]-amino-6-methylpyridineの合成とスクリーニング
- 鎮痛作用物質5-Aminomethylsalicylic Acidの合成研究
- Studies on Analgesics of Aniline Series. III. Preparation and Properties of N, N-Dialkyl 3-(Substituted anilino) butyramide Series
- Studies on Analgesics of Aniline Series. II. Preparation and Properties of N-Alkyl or N, N-Dialkyl 3-(N'-Acyl- or N'-Benzyl-substituted anilino) propionamide Series and N-Alkyl or N, N-Dialkyl 3-(Substituted anilino) propylamine Series
- Studies on Analgesics of Aniline Series. I. Preparation and Properties of β-Alaninamide Series
- Studies on Steroids. III. The Preparation of Steroid-21-yl-glucopyranosiduronamides.
- Studies on Antiviral Agents. I. Relationship between Chemical Reactivity of Sulfhydryl Reagents and Their Inactivating Activity of Adenovirus Type 5
- D-Glucuronolactone Derivatives. VII. Synthesis of Anomeric 1-Deoxy-1-halogeno-2,5-di-O-acyl-D-glucofuranurono-γ-lactones
- Ruthenium Tetroxide Oxidation of N-Alkyllactams(Organic,Chemical)
- Ruthenium Tetroxide Oxidation of 1-Azabicycloalkan-2-ones
- Studies on Antiviral Agents. III. Synthesis of Tenuazonic Acid Derivatives.
- Studies on Oxidized Starch Sulfates for Medical Purposes. I. Synthesis of Sulfates of Oxidized Starch and its Derivatives.
- Studies on Sulfonylurea Derivatives. III. The Infrared Spectra of 1-p-Tolylthio-3-alkylureas and Corresponding Sulfonyl Compounds.
- 気軽に立ち寄れる会館に(新薬学会館に望む)
- The Selective Dealkylation of Mixed Esters of Phosphoric Acid and Phenylphosphonic Acid Using Cation Exchange Resin
- Reaction of Amino Acids with Alkyl p-Toluenesulfonates
- Reaction of Carboxylic Acid Esters with p-Toluenesulfonic Acid
- Reaction of Ethyl Acetoacetate with p-Toluenesulfonic Acid : Formation of Ethyl Isodehydroacetate and/or Ethyl p-Toluenesulfonate
- Derivees des Pyrimidines. II. Synthese des Alcocy-2-Pyrimidyl-4)-N^1-Sulfanilamides
- Pyrimidine Derivatives. I. Synthesis of a New Series of Sulfanilamides having Dialkylamino Groups in the Pyrimidine Nucleus
- Pyridazines. XI. Pyrido[2,3-d]pyridazines. II
- Pyridazine Derivatives. VIII. Pyrido[2,3-d]pyridazines. I.
- The Syntheses of Some Aminomethylindoles
- 柴胡桂枝湯の神経薬理学的研究(第2報)
- 柴胡桂枝湯の神経薬理学的研究(第1報)
- Electronic Structure and Local Anesthetic Activity of 2-Diethylaminoacetanilide Derivatives
- Electronic Structure and Antibacterial Activity of Nitrofuran Derivatives
- 柴胡桂枝湯の神経薬理学的研究(第4報) : 煎剤およびエキス中の抗PTZ作用生薬の成分含量
- 柴胡桂枝湯の神経薬理学的研究(第3報) : 神経線維に対する麻酔作用
- Pyridazine Derivatives. IV. The Structures of Aminopyridazines.
- Pyridazine Derivatives. II. Infrared Spectra of O-, N-Mono- and O, N-Dibenzyl Compounds of Maleic Hydrazide.