Studies on Steroids. I. The Preparation and Properties of 17β-(N-Substituted 2-Amino-4-thiazolyl)-androst-4-en-3-one Series.
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概要
- 論文の詳細を見る
17β-(2-alkylamino-(or 2-arylamino- or 2-N, N-alkylarylamino-)-4-thiazolyl) androst-4-en-3-one derivatives were prepared from Reichstein's compound S 21-iodide, cortisone 21-iodide and desoxycorticosterone 21-iodide or corresponding 21-mesylate with N-alkylthiourea, N-arylthiourea or N, N-alkylarylthiourea respectively. Some of these compounds were found to have a digitalis-like properties (cardiac glucoside properties) as a result of pharmacological test.
- 社団法人日本薬学会の論文
- 1963-05-25
著者
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高村 圭一
中外製薬株式会社綜合研究所
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磯野 千冬
中外製薬綜研
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磯野 千冬
中外製薬株式会社綜合研究所
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高村 圭一
Research Laboratory, Chugai Pharmaceutical Co., Ltd.
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磯野 千冬
Research Laboratory, Chugai Pharmaceutical Co., Ltd.
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新田 義博
Research Laboratory, Chugai Pharmaceutical Co., Ltd.
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高久 栄
Research Laboratory, Chugai Pharmaceutical Co., Ltd.
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高久 栄
中外製薬綜研
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高久 栄
中外製薬株式会社綜合研究所
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新田 義博
School Of Pharmacy Hokuriku University
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