Studies on Mesoionic Compounds. XII. Synthesis of 1,2,3-Thiadiazolium-4-aminide Derivatives and Their Characterization
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概要
- 論文の詳細を見る
New mesoionic heterocycles, 1,2,3-thiadiazolium-4-ethoxycarbonylaminides (9 and 10), were prepared by alkylation of 1,2,3-thiadiazoles (5) followed by treatment with base. Compound (9) was hydrolyzed to the hydrochloride of the corresponding 4-imine derivative (13), which was converted to the 4-oxo analog (16) via N-nitrosation.
- 社団法人日本薬学会の論文
- 1981-06-25
著者
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森田 光
Central Research Laboratories Zeria Pharmaceutical Co. Ltd.
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増田 克忠
Faculty of Pharmaceutical Sciences, Toyama Medical Pharmaceutical University
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安立 準
Faculty of Pharmaceutical Sciences, Toyama Medical Pharmaceutical University
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森田 光
Faculty of Pharmaceutical Sciences, Toyama Medical Pharmaceutical University
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野村 敬一
Faculty of Pharmaceutical Sciences, Toyama Medical Pharmaceutical University
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野村 敬一
Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University
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増田 克忠
Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University
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安立 準
Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University
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