Sur les Possibilites de Formation de Pyrimidines a partir de la Dibromo-3,4 dihydro-3,4 coumarine
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概要
- 論文の詳細を見る
Reactions of 3,4-dibromo-3,4-dihydrocoumarin (3) with acetamidine and benzamidine gave 6-(2-hydroxyphenyl)-4-oxo-3,4-dihydropyrimidines (1a and 1b) having in the 2-position the methyl and phenyl substituents, respectively. In these reactions, the coumarin 3 was converted in the first place into 3-bromocoumarin (4) which was then transformed to the pyrimidines 1a and 1b. The coumarin 4 did not undergo the Perkin rearrangement with amidines.
- 社団法人日本薬学会の論文
- 1982-12-25
著者
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森田 光
Central Research Laboratories Zeria Pharmaceutical Co. Ltd.
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高田 純
北里大(薬)
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高木 要
Laboratoire de Chimie, Zeria Pharmaceutical Co., Ltd.
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森田 光
Laboratoire de Chimie, Zeria Pharmaceutical Co., Ltd.
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長原 勝彦
Faculte des Sciences Pharmaceutiques, Universite Kitasato
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高田 純
Faculte des Sciences Pharmaceutiques, Universite Kitasato
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長原 勝彦
Faculte Des Sciences Pharmaceutiques Universite Kitasato
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高木 要
Central Research Laboratories, Zeria Pharmaceutical Co., Ltd.
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高木 要
Central Research Laboratories Zeria Pharmaceutical Co. Ltd.
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