The Reaction of α, β-Unsaturated Ketones with Azides. III.

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概要

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• The reaction of seven kinds of conjugated bicycloalkenones (I, III, V, VII, IX, XV and XX) with hydrazoic acid were studied. From compounds (I, III, V and VII), enone type lactams were obtained and from compounds (IX, XV and XX), α, β-unstaturated α-aminoketones were obtained. The three types of reaction products (a) lactams, b) α, β-unsaturated α-aminoketones and c) β-diketones) were observed from present and previous results. The correlation between the structure of α, β-unsaturated ketone and the reaction product was discussed.

• 公益社団法人日本薬学会の論文
• 1969-08-25

著者

• 南 法夫

  Eisai Tsukuba Research Laboratories

• 野村 敬一

  Faculty of Pharmaceutical Sciences, Toyama Medical Pharmaceutical University

• 野村 敬一

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

• 松山 稔

  Faculty Of Pharmaceutical Sciences University Of Toyama

• 三橋 監物

  Faculty of Pharmaceutical Sciences, University of Toyama

• 南 法夫

  Research Laboratories Eisai Co. Ltd.

• 南 法夫

  Faculty of Pharmaceutical Sciences, University of Toyama

• 三橋 監物

  Faculty Of Pharmaceutical Sciences Josai University

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