AN EFFICIENT 3(C)-ACYLATION OF TETRAMIC ACIDS INVOLVING ACYL MIGRATION OF 4(O)-ACYLATES(Communications to the Editor)

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概要

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• 3(C)-Acylation of 3-unsubstituted tetramic acids with carboxylic acid has been achieved by two sequential reactions in one flask: (1) 4(O)-acylation in. the presence of DCC.and a catalytic amount of DMAP, and (2) 4(O)-}3(C) acyl-migration promoted by adding Et_3N.

• 公益社団法人日本薬学会の論文
• 1987-10-25

著者

• 野村 敬一

  Faculty of Pharmaceutical Sciences, Toyama Medical Pharmaceutical University

• 野村 敬一

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

• 吉井 英一

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

• 吉井 英一

  富山医科薬科大学薬学部

• 堀 耕造

  Faculty of Pharmaceutical Sciences, Toyama Medical and Pharmaceutical University

• 荒井 幹雄

  Faculty of Pharmaceutical Sciences, Toyama Medical and Pharmaceutical University

• 荒井 幹雄

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

• 堀 耕造

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

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