N-モノ置換Diphenylphosphinamide類のアルキル化反応

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概要

• 論文の詳細を見る

• A facile preparative method for N, N-disubstituted diphenylphosphinamides was developed. Treatment of N-alkyl (or phenyl) diphenylphosphinamides with a slight excess of sodium hydride followed by a reaction with alkyl halides produced the corresponding N, N-disubstituted derivatives in a fair yield. It is suggested that this method of N-alkylation provides a potentially useful means for the conversion of primary amines to secondary amines.

• 社団法人日本薬学会の論文
• 1977-09-25

著者

• 小泉 徹

  富山医科薬科大学薬学部薬化学

• 小泉 徹

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

• 小林 恵子

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

• Koizumi T

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

• 小林 恵子

  富山大学薬学部

• 小泉 徹

  富山大学薬学部

• 吉井 英一

  富山大学薬学部

• 吉井 英一

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

• 吉井 英一

  富山医科薬科大学薬学部

• Koizumi Toru

  Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University

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