SUCCESSFUL ASYMMETRIC DIELS-ALDER APPROACH TO OPTICALLY ACTIVE C-NUCLEOSIDES. ENANTIOSELECTIVE TOTAL SYNTHESIS OF D-SHOWDOMYCIN AND D-2,5-ANHYDROALLOSE DERIVATIVES(Communications to the Editor)
スポンサーリンク
概要
- 論文の詳細を見る
Using an asyntmetric Diels-Alder reaction of (S)_S-3-(2-pyridyl-sulfinyl)acrylate with furan, a highly enantioselective synthesis of a common key intermediate (+)-(1) was achieved, and this was successfully converted to C-nueleosides, D-showdomycin (2) and D-3, 4-O-isopropylidene-2,5-anhydroallose (3).
- 社団法人日本薬学会の論文
- 1987-01-25
著者
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高山 広光
Faculty of Pharmaceutical Sciences, Chiba University
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小泉 徹
富山医科薬科大学薬学部薬化学
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小泉 徹
Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University
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伊与部 亮
Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University
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高山 広光
Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University
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Koizumi T
Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University
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小泉 徹
Department Of Synthetic Organic Chemistry:faculty Of Pharmaceutical Sciences Toyama Medical And Phar
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Koizumi Toru
Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University
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高山 広光
Faculty Of Pharmaceutical Sciences Chiba University
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