Synthesis of α-(Methylthio)arylacetamides and Their Conversion into Some Biologically Active Arylethylamines

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概要

• 論文の詳細を見る

• A series of (methylsulfinyl)acetamides 4 reacted with electron-rich arenes in the presence of p-toluenesulfonic acid to give α-(methylthio)arylacetamides 5,6,and 7,some of which were transformed into biologically active arylethylamines such as (±)-macromerine.

• 社団法人日本薬学会の論文
• 1989-12-25

著者

• 池田 正澄

  Kyoto Pharmaceutical University

• 池田 正澄

  京都薬科大学

• 石橋 弘行

  Kyoto Pharmaceutical University

• 石橋 弘行

  金沢大学薬学部

• 石橋 弘行

  京都薬科大学

• 三木 裕美子

  Kyoto Pharmaceutical University

• 池田 美朗

  Kyoto Pharmaceutical University

• 喜里山 暁子

  Kyoto Pharmaceutical University

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