Enantio- and Diastereoselective Synthesis of N-[(1R, 2R, 3R, 4R)-2,3-Diacetoxy-4-(acetoxymethyl)cyclopentyl]acetamide, a Synthetic Key Intermediate of (+)-Cyclaradine
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概要
- 論文の詳細を見る
Enantio- and diastereoselective synthesis of N-[(1R, 2R, 3R, 4R)-2,3-diacetoxy-4-(acetoxymethyl)cyclopentyl]-acetamide 1,a synthetic key intermediate of (+)-cyclaradine, has been achieved by using enzyme-catalyzed asymmetric hydrolysis and subsequent modification of a functional group.
- 公益社団法人日本薬学会の論文
- 1998-05-15
著者
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田中 正一
Graduate School Of Pharmaceutical Sciences Kyushu University
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TANAKA Masakazu
Faculty of Bioscience, Nagahama Institute of Bio-Science and Technology
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Tanaka M
Faculty Of Pharmaceutical Sciences Tokushima Bunri University
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Hayashi Masaki
Faculty of Horticulture, Chiba University
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SUEMUNE HIROSHI
Faculty of Pharmaceutical Sciences, Kyushu Uinversity
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NORIMINE Yoshihiko
Faculty of Pharmaceutical Sciences, Kyushu University
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Suemune H
Graduate School Of Pharmaceutical Sciences Kyushu University
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Suemune Hiroshi
Faculty Of Pharmaceutical Sciences Kyushu Uinversity
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Norimine Yoshihiko
Faculty Of Pharmaceutical Sciences Kyushu University
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Hayashi M
Faculty Of Pharmaceutical Sciences Kyushu University
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