Pyrrolidine-Forming 1,3-Dipolar Cycloaddition of N-(Phenylthiomethyl)-α-amino Acid Esters

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概要

• 論文の詳細を見る

• The sodium hydride-aided reaction of N-(phenylthiomethyl)-α-amino acid esters with α, β-unsaturated carboxylates results in a pyrrolidine-forming 1,3-dipolar cycloaddition. Thus, a new route to pyrrolidines, pyrrolizidines, and indolizidines has been provided.

• 社団法人日本薬学会の論文
• 1986-03-25

著者

• 今井 信行

  Shizuoka College Of Pharmacy

• 関屋 実

  School Of Pharmaceutical Sciences University Of Shizuoka

• 寺尾 良保

  Shizuoka College of Pharmacy

• 関屋 実

  Shizuoka College of Pharmacy

• 寺尾 良保

  School Of Pharmaceutical Sciences University Of Shizuoka

• 阿知波 一雄

  Shizuoka College of Pharmacy

• 根本 まり

  Shizuoka College of Pharmacy

関連論文

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• Reactions of 2,2-Dichlorovinyl and 2,2-Dichlorovinylidene Sulfides with Butyllithium
• Thermal Rearrangements of Allyl 2,2-Dichloro-, 1,2-Dichloro- and 1,2,2-Trichloro-substituted Vinyl Sulfides
• Novel Rearrangements of α-N-Alkylamido-substituted Sulfides and Sulfones
• Syntheses and Reactions of Phenylthio-and Propylthioacetylenic Compounds
• Enantioface-Differentiating Epoxidation of Alkylidenemalononitriles with Molecular Oxygen, catalyzed by Chiral Tertiary Amines
• Formic Acid Reduction. XXVIII. Kinetic Studies on the Formic Acid Reduction of 1,1'-Benzylidenedipiperidine
• A New Insertion Reaction of Diazoalkanes with Dialkylaminomethyl Esters of Dialkyldithiocarbamic Acid and of Ethylxanthic Acid
• Chlorinolyses of Alkyl (or Aryl) Phthalimidomethyl Sulfoxides with Sulfuryl Chloride, Chlorine and Thionyl Chloride
• Nucleophilic Substitution of Alkyl (or Aryl) Imidomethyl Sulfones. A New Convenient Synthesis of Alkane (or Arene) sulfinates
• Decarboxylation Reaction. VIII. Reaction of Electron-deficient Carbon-Carbon Double Bonds with Trichloroacetic Acid. A Unique 1,1-Dichlorocyclopropane Formation through β-Trichloromethylation
• Formic Acid Reduction. XXVI. α, β-Reduction of Conjugated Nitriles with Formic Acid
• Decarboxylation Reactions. V. Reaction of N-Benzylideneanilines with Propiolic Acid
• Formic Acid Reduction. XXIV. Path of the Reductive Fission of the Centered β-Carbon Bond of Alkylidenebisketones
• Formic Acid Reduction. XXIII. Kinetic Studies on the Formic Acid Reduction of Carbon-Carbon Double Bond Adjacent to Carbonyl
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• オクテット
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• Synthesis of N-(Alkylaminomethyl) amides

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