Trifluoromethanesulfonic Acid-Promoted Reaction of Hexahydro-1,3,5-triazines.Introduction of a Secondary Aminomethyl Grouping into Carboxylates at the α-Position through Ketene Silyl Acetals

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概要

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• Introduction of the secondary aminomethyl grouping RNHCH_2 into carboxylates at the α-position has been achieved by reaction of hexahydro-1,3,5-triazines with ketene silyl acetals in the presence of a catalytic amount of trifluoromethanesulfonic acid.

• 社団法人日本薬学会の論文
• 1986-04-25

著者

• 関屋 実

  School Of Pharmaceutical Sciences University Of Shizuoka

• 関屋 実

  Shizuoka College of Pharmacy

• 池田 潔

  Shizuoka College Of Pharmacy

• 阿知波 一雄

  Shizuoka College of Pharmacy

• 池田 かおり

  Developmental Research Laboratories Shionogi & Co. Ltd.

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