Reaction of 1-Pyrrolidino-1-cyclohexene with Imidoyl Chlorides and a Route to Producing Phenanthridines

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概要

• 論文の詳細を見る

• Reaction of 1-pyrrolidino-1-cyclohexene with N-arylbenzimidoyl chlorides has been successfully performed to result in introduction of benzimidoyl groupings at β-carbon of the enamine. Easy hydrolysis of enamine moiety of these products provides an effective means of preparation of mono-anils of 2-benzoylcyclohexanone, from which several phenanthridine derivatives have been newly obtained by action of polyphosphoric acid.

• 公益社団法人日本薬学会の論文
• 1975-06-25

著者

• 関屋 実

  School Of Pharmaceutical Sciences University Of Shizuoka

• 関屋 実

  Shizuoka College of Pharmacy

• 森本 俊明

  Shizuoka College of Pharmacy

関連論文

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