Azole Series. I. Reaction of 2-(Acylamino)thioacetamides, leading to 5-Aminothiazoles and to Thiazolo[5,4-d]pyrimidines.
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Formation of 5-acetamido-substituted thiazoles was found to be readily effective on heating 2-(acylamino)thioacetamides with acetic anhydride. In additon, preparation of some starting 2-(acylamino)thioacetamides is described and 5-acetamidothiazole-4-carboxamides obtained by the thiazole formation reaction were led to some thiazolo[5,4-d]pyrimidines.
- 公益社団法人日本薬学会の論文
- 1965-11-25
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関連論文
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