Synthesis of Pyridinium Dinitrobenzyl Sulfates and Potassium (Dinitrobenzyl β-D-Glucopyranosid)Uronates
スポンサーリンク
概要
- 論文の詳細を見る
Sulfates and glucuronides of 2,4-dinitrobenzyl alcohol 1a and 2,6-dinitrobenzyl alcohol 1b, which are major or putative metabolites of 2,4-dinitrotoluene (2,4-DNT) and 2,6-dinitrotoluene (2,6-DNT), were synthesized from 1a and 1b by reaction with pyridinium sulfonate and methyl (2,3,4-tri-O-acetyl-α-D-glucopyranosyl)uronate bromide 3,respectively, as their pyridinium salts (2a, 2b) and potassium salts (6a, 6b). These conjugates are important for the study of the carcinogenicity of 2,4-DNT and 2,6-DNT.
- 公益社団法人日本薬学会の論文
- 1998-01-15
著者
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Inoue M
Lab. Of Medicinal Resources School Of Pharmacy Aichi Gakuin Univ.
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DOHRIN Masahiro
Faculty of Pharmaceutical Sciences, Toyama Medical & Pharmaceutical University
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Inoue M
Laboratory Of Pharmacognosy Graduate School Of Pharmaceutical Sciences Nagoya City University
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KOZUKA HIROSHI
Faculty of Pharmaceutical Sciences, Toyama Medical and Pharmaceutical University
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MORI Masa-aki
Department of Health Sciences, School of Medicine, Kyushu University
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Inoue M
Nagoya‐city Univ. Aichi Jpn
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Kozuka H
Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University
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Mori Masa-aki
Department Of Health Sciences School Of Medicine Kyushu University
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Sayama M
Department Of Material Systems Engineering And Life Science Faculty Of Engineering Toyama University
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Mori Masa-aki
School of Health Sciences, Kyushu University
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Shoji Miki
Faculty of Medicine, Toyama Medical and Pharmaceutical University
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SAYAMA Michio
Toyama Medical and Pharmaceutical University
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INOUE Masami
Toyama Medical and Pharmaceutical University
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Dohrin Masahiro
Faculty Of Pharmaceutical Sciences Toyama Medical And Pharmaceutical University
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Shoji Miki
Faculty Of Medicine Toyama Medical And Pharmaceutical University
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Kozuka Hiroshi
Faculty Of Medical Sciences Toyama Medical And Pharmaceutical University
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Mori Masaaki
School of Health Sciences, Kyushu University
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