A Facile Method for the Stereoselective Horner-Wadsworth-Emmons Reaction of Aryl Alkyl Ketones

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概要

• 論文の詳細を見る

• Excellent Z or E selectivity was observed in the Horner-Wadsworth-Emmons (HWE) reactions of methyl bis(2,2,2-trifluoroethyl)phosphonoacetate or ethyl 2-fluoro-2-diethylphosphonoacetate with aryl alkyl ketones bearing substituents on an aromatic moiety employing Sn(OSO_2CF_3)_2 in the presence of N-ethylpiperidine.

• 公益社団法人日本薬学会の論文
• 2002-05-01

著者

• Yokoyama Kazumasa

  Central Research Laboratories Green Cross Corporation Ltd.

• SHIRO Motoo

  Rigaku Corporation X-ray Research Laboratory

• Shiro Motoo

  Rigaku Corporation

• Shiro M

  Rigaku Corp. Tokyo

• NAGAO Yoshimitsu

  Faculity of Pharmaceutical Sciences, The University of Tokushima

• SANO Shigeki

  Faculty of Pharmaceutical Sciences, The University of Tokushima

• 佐野 茂樹

  Graduate School Of Pharmaceutical Sciences The University Of Tokushima

• 佐野 茂樹

  徳島大学薬学部

• 長尾 善光

  Graduate School Of Pharmaceutical Sciences The University Of Tokushima

• 長尾 善光

  徳島大学薬学部

• YOKOYAMA Kenji

  Faculty of Pharmaceutical Sciences, The University of Tokushima

• Nagao Y

  Faculty Of Pharmaceutical Sciences The University Of Tokushima

• Nagao Yoshimitsu

  Faculity Of Pharmaceutical Sciences The University Of Tokushima

• Yokoyama K

  Showa Pharmaceutical University

• Shiro M

  Rigaku Corporation

• Suzuki Mitsuko

  Institute For Chemical Research Kyoto University

• Masuoka S

  Takara Agri Co. Ltd.

• Yamanouchi K

  Faculty Of Pharmaceutical Sciences The University Of Tokushima

• Shiro Motoo

  Rigaku Co.

• Shiro Motoo

  Shionogi Research Laboratry Shionogi & Co. Ltd.

• Mito S

  Institute For Chemical Research Kyoto University

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