A facile synthesis of 3-hydroxymethyl- and 3-formylindoles from o-nitrotoluene.

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概要

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• A synthesis of 3-hydroxymethyl- and 3-formylindoles has been performed by manipulation of the side chain of 3-hydroxymethylindoline derived from <I>o</I>-nitrotoluene. Electro-reductive cyclization of 2-(2-nitro-phenyl)-1,3-bis(methylsulfonyloxy)propane to 3-(benzyloxymethyl)indole, is also discussed.

• 公益社団法人 日本化学会の論文

著者

• Okamoto Koichi

  Deparment Of Neurology Gunma University School Of Medicine

• Torii Sigeru

  Department Of Applied Chemistry Faculty Of Engineering Okayama University

• Murakami Yasuo

  Department Of Anesthesiology Saitama Medical School

• Tanaka Hideo

  Department Of Applied Chemistry Faculty Of Engineering Okayama University

• Murakami Yasuo

  Department of Industrial Chemistry, School of Engineering, Okayama University

• Aizawa Takao

  Department of Applied Chemistry, Faculty of Engineering, Okayama University

• Aizawa Takao

  Department of Industrial Chemistry, School of Engineering, Okayama University

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