An Efficient Method for Preparing gem-Dimethylcyclopropanes from gem-Dibromocyclopropanes(Organic,Chemical)

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概要

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• Reaction of gem-dibromocyclopropanes (1) with a higher-order organocuprate prepared from cuprous thiocyanate and methyllithium, followed by the addition of methyl iodide in situ, readily afforded dimethylcyclopropanes (2) in good to excellent yields regardless of the functional group in 1.

• 社団法人日本薬学会の論文
• 1987-12-25

著者

• 小川 和宏

  Faculty Of Pharmaceutical Sciences Kyoto University

• 原山 尚

  Faculty of Pharmaceutical Sciences, Chiba University

• 福士 英人

  Faculty of Pharmaceutical Sciences, Kyoto University

• 荒谷 哲也

  Faculty of Pharmaceutical Sciences, Kyoto University

• 曽根原 聡

  Faculty of Pharmaceutical Sciences, Kyoto University

• 米田 文郎

  Faculty of Pharmaceutical Sciences, Kyoto University

• 曽根原 聡

  京都大学薬学部

• 荒谷 哲也

  Faculty Of Pharmaceutical Sciences Kyoto University

• 原山 尚

  Faculty Of Pharmaceutical Sciences Kyoto University

• 福士 英人

  Pharamaceutical Research Laboratories I Pharmaceutical Research Division Takeda Chemical Industries

• 米田 文郎

  Faculty Of Pharmaceutical Sciences Kyoto University

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