1,3-ジメチルチミンエポキシドとアミン類との反応における溶媒効果(有機化学)
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概要
- 論文の詳細を見る
The solvent effect in reaction of 1,3-dimethylthymine epoxide with amines was investigated. The results are summarized in Table I, indicating that the ratio of formation of cis product (2) increases as a solvent becomes more polar. This suggests that a polar solvent stabilizes an ionic intermediate (1B), which reacts with amine to afford the cis product selectively.
- 公益社団法人日本薬学会の論文
- 1986-11-25
著者
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原山 尚
京都大学薬学部
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米田 文郎
京都大学薬学部
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原山 尚
Faculty Of Pharmaceutical Sciences Kyoto University
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柳田 玲子
京都大学薬学部
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米田 文郎
Faculty Of Pharmaceutical Sciences Kyoto University
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飯尾 公美子
京都大学薬学部
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