α-アドレナリン遮断作用を有するアポガランタミン類似体の合成(第4報)光化学閉環による合成その2
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概要
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The apogalanthamine analogs, 10,11-methylenedioxy-(1) and 10,11-dimethoxy-5,6,7,8-tetrahydrodibenz [c, e] azocine (2), as α-adrenergic blocking agents were synthesized by photolysis of N-benzyl-2-bromo-4,5-methylenedioxy-(9) and N-benzyl-2-bromo-4,5-dimethoxy-β-phenethylamine (10). 2,3-Methylenedioxy-(3) and 2,3-dimethoxy-5,6,7,8-tetrahydrodibenz [c, e] azocine (4), were also prepared by photolysis of N-(2-bromo-4,5-methylenedioxybenzyl)-(11) and N-(2-bromo-4,5-dimethoxybenzyl)-β-phenethylamine (12).
- 1978-02-25
著者
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小林 茂
Faculty Of Home Economics Shikoku University
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木原 勝
徳島大学薬学部
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木原 勝
Faculty Of Pharmaceutical Sciences The University Of Tokushima
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小林 茂
徳島大学薬学部
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中内 康起
徳島大学薬学部
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