Syntheses of Apogalanthamine Analogs as α-Adrenergic Blocking Agents. III. 5,6,7,8-Tetrahydrodibenz [c, e] azocine and Its 6-Substituted Derivatives
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概要
- 論文の詳細を見る
The apogalanthamine analogs, 5,6,7,8-tetrahydrodibenz [c, e] azocine (10) and its Nsubstituted derivatives (11-15) were synthesized. Boron tribromide was found to be effective for cleavage and bromination of the lactone ring in diphenide (25). This is the first time it has been employed as a cleaving and brominating agent for a lactone.
- 公益社団法人日本薬学会の論文
- 1978-02-25
著者
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小林 茂
Faculty Of Home Economics Shikoku University
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木原 勝
Faculty Of Pharmaceutical Sciences The University Of Tokushima
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小林 茂
四国女子大学家政学部
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峯尾 哲
Faculty Of Pharmaceutical Sciences Tokushima University
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