Syntheses of Apogalanthamine Analogs as α-Adrenergic Blocking Agents. VIII. Syntheses of 4- and 9-Bromo-5,6,7,8-tetrahydrodibenz [c, e] azocines and Their Methylenedioxy Derivatives
スポンサーリンク
概要
- 論文の詳細を見る
The apogalanthamine analogs 4- and 9-bromo-5,6,7,8-tetrahydrodibenz [c, e] azocines (5a and 6a) and their methylenedioxy derivatives (5b and 6b) were prepared by photolysis of the hydrochlorides of the respective N-benzyl-β-phenethylamines (8a, b and 9a, b) substituted with both iodine and bromine atoms. The dibenz [c, e] azocines 6a and 6b were also obtained by thermal syntheses from the biphenyl compounds 17a and 17b, respectively.
- 社団法人日本薬学会の論文
- 1985-03-25
著者
-
小林 茂
Faculty Of Home Economics Shikoku University
-
木原 勝
Faculty Of Pharmaceutical Sciences The University Of Tokushima
-
三宅 美行
Faculty of Pharmaceutical Sciences, Tokushima University
-
飯富 守夫
Faculty of Pharmaceutical Sciences, Tokushima University
-
三宅 美行
Faculty Of Pharmaceutical Sciences Tokushima University
-
飯富 守夫
Faculty Of Pharmaceutical Sciences Tokushima University
関連論文
- α-アドレナリン遮断作用を有するアボガランタミン類似体の合成(第7報)2-Iodo-N-(2-iodobenzyl)-β-phenethylamineの光化学閉環
- α-アドレナリン遮断作用を有するアポガランタミン類似体の合成(第4報)光化学閉環による合成その2
- Alkaloidal Constituents of Leucojum autumnale L. (Amaryllidaceae)
- Regioselective Cleavage Reaction of the Aromatic Methylenedioxy Ring. VI. Synthesis of Phenothiazine Analogues by Using the Cleavage Reaction with Sodium Methoxide-Thiols in Dimethyl Sulfoxide and Evaluation of Their Biological Activities
- Isolation and Structure Elucidation of a Novel Alkaloid, Incartine, a Supposed Biosynthetic Intermediate, from Flowers of Lycoris incarnata
- Regioselective cleavage Reaction of the Aromatic methylenedioxy Ring. V. Cleavage with Sodium Alkoxides-Alcohols, Potassium tert-Butoxide-Alcohols, Dimsyl Anion-Methyl Alcohol, Metallic Sodium-Alcohols, and Sodium Cyanide in Dipolar Aprotic Solvents
- Alkaloidal Constituents of the Flowers of Lycoris radiata HERB. : Amaryllidaceae
- Synthesis of Apogalanthamine Analogues as α-Adrenergic Blocking Agents. XIII. Syntheses of Phenolic 8-Hydroxy-5,6,7,8-tetrahydrodibenz[c, e]azocines
- Syntheses of Apogalanthamine Analogues as α-Adrenergic Blocking Agents. XII. : Syntheses and Stereochemistry of Methoxy and Methylenedioxy Derivatives of 8-Hydroxy-5,6,7,8-tetrahydrodibenz-[c, e]azocines
- Alkaloidal Constituents of Hymenocallis rotata HERB. (Amaryllidaceae)(Organic,Chemical)
- Structures of Acid B and Related Compounds, Oxidation Products of Lycoramine
- Structure and Synthesis of Acid A, an Oxidation Product of Lycoramine
- Iridoid Glucosides from Lamium amplexicaule
- Alkaloidal Constituents of Leucojum asetivum L. (Amaryllidaceae)
- Studies on Constituents of Bignoniaceae Plants. IV. Isolation and Structure of a New Iridoid Glucoside, Campsiside, from Campsis chinensis
- Syntheses of Apogalanthamine Analogs as α-Adrenergic Blocking Agents. VIII. Syntheses of 4- and 9-Bromo-5,6,7,8-tetrahydrodibenz [c, e] azocines and Their Methylenedioxy Derivatives
- Alkaloidal Constituents of Crinum latifolium and Crinum bulbispermum (Amaryllidaceae)
- ANTIFEEDANTS FOR THE LARVAE OF THE YELLOW BUTTERFLY, EUREMA BECABE MANDARINA, IN LYCORIS RADIATA
- Cleavage of the Methylenedioxy Ring. III. Cleavage with Sodium Benzyloxide in Dimethyl Sulfoxide
- Isolation of O-Demethyllycoramine from Bulbs of Lycoris radiata HERB.
- Transformation of Tazettine to Pretazettine
- 四年生の講座配属について(四年生の講座配属)
- Synthesis and Enantioselectivity of Optically Active 1- and 3-Substituted 4-Phenyl-1,2,3,4-tetrahydroisoquinolin-4-ols and Related Compounds as Norepinephrine Potentiators
- New Norepinephrine Potentiators : Synthesis and Structure-Activity Relationships of a Series of 4-Phenyl-1,2,3,4-tetrahydroisoquinolin-4-ols
- Isolation of N-Demethylgalanthamine from the Bulbs of Crinum asiaticum L. var. japanicum BAKER (Amaryllidaceae)
- Alkaloids of the Amaryllidaceae. A New Alkaloid, Sanguinine, from Lycoris sanguinea MAXIM. var. Kiushiana MAKINO, and Pretazettine from Lycoris radiata HERB.
- Galanthamine Chemistry. V. Formation of Hydroxyapogalanthamine from Galanthaminone and the Synthesis of its Trimethyl Ether.
- Photochemical Syntheses of Apogalanthamine Analogs as α-Adrenergic Blocking Agents
- Syntheses of Apogalanthamine Analogs as α-Adrenergic Blocking Agents
- ジフェン酸モノメチルエステル誘導体の合成 その2
- Studies on the α-Adrenolytic Activities of Apogalanthamine Analogs
- 2′-Bromomethyl-2-biphenylcarbaldehydeとシアン化ナトリウムとの反応
- Synthesis of 6-(β-Bromoethyl)-10,11-methylenedioxy-5,6,7,8-tetrahydrodibenz-[c, e]azocine (DA-VIII-MBr) as a New Specific α-Adrenergic Blocking Agent
- Synthesis of 2'-Cyanomethyl-2-biphenylcarboxylic Acid
- Studies on the Syntheses of Benzoheterocyclic Compounds. VI. Diphenide and Its Methoxyl Derivatives
- Lycoris Alkaloids. XXIV. : Isolation and Characterization of Lycoremine.
- 駆虫薬の合成研究 第6・7報
- ハロゲン置換N-Benzyl-β-phenethylamine誘導体の光化学反応について
- Syntheses of Apogalanthamine Analogs as α-Adrenergic Blocking Agents. III. 5,6,7,8-Tetrahydrodibenz [c, e] azocine and Its 6-Substituted Derivatives
- Syntheses of Methylenedioxydiphenides and Dimethoxydiphenides
- Isolation of Clivacetine from Clivia miniata REGEL. (Amaryllidaceae)
- Isolation of Carinatine and Pretazettine from the Bulbs of Zephyranthes carinate HERB. (Amaryllidaceae)
- Synthesis of optically Active Deoxytazettine Neomethine
- Cleavage of the Methylenedioxy Ring. II. Cleavage with Sodium Phenoxide and Methoxide in Dimethyl Sulfoxide
- Cleavage of the Methylenedioxy Group with Sodium Methoxide in Dimethyl Sulfoxide
- Alpha-adrenolytic Activities of N-Benzyl-β-phenethylamine Derivatives on Isolated Smooth Muscles